欧美高清

欧美高清-GSKOur Publications

Over 180 primary peer-reviewed research papers have been published to date, with many in high impact journals, including Angew. Chem., Int. Ed.; J. Am. Chem. Soc.; Chem. Sci.; ACS Chem. Biol.; ACS Catal.; and J. Med. Chem.  Additionally, 26 patents have been filed based on research carried out as part of our collaborative projects.

Across the programme, research projects are carefully selected to advance innovation and understanding in areas of science that are relevant to the pharmaceutical industry in general or GSK in particular.

Collaborative Research Papers

182. . Chelsea D. Grace, John A. Murphy, and Simon M. Nicolle, Chem. Eur. J., 2025, 31, e01908.

181. . Aidan McKeown, Jonathan A. Taylor, Laura C. Paterson, David M. Lindsay, and William J. Kerr, Adv. Synth. Catal., 2025, e70168.

180. . Natasha Sanjrani, Damien E. Coupry, Peter Pogany, David S. Palmer, and Stephen D. Pickett, J. Chem. Inf. Model, 2025, ASAP article. DOI:

179. . Caitlin Fawcett, Joe Watson, Stephen Richards, Alfred E. Doherty, Hikaru Seki, Elizabeth A. Love, Charlotte H. Coles, Diane M. Coe, and Craig Jamieson, Bioconjugate Chem., 2025, 36, 1054-1065.

178. . Luke Chen, James Thompson, and Craig Jamieson, Adv. Synth. Catal., 2025, accepted article. DOI: .

177. . James Lodge, Lewis Kajtar, Rachel Duxbury, David Hall, Glenn A. Burley, Joanna Cordy, James W. T. Yates, and Zahra Rattray, mAbs, 2025, 17, 2459795.

176. . Rebecca Stevens, Harry E. P. Palmer, Afjal H. Miah, and Glenn A. Burley, J. Org. Chem., 2025, 90, 2192-2200.

175. . Harry Wilders, George Biggs, Sam M. Rowe, Emma E. Cawood, Ioannis G. Riziotis, Alan R. Rendina, Emma K. Grant, Jonathan Pettinger, David J. Fallon, Mark Skehel, David House, Nicholas C. O. Tomkinson, and Jacob T. Bush, Angew. Chem. Int. Ed., 2025, 64, e202418314.

174. . Rebecca Stevens, Harry J. Shrives, Jenni Cryan, Diana Klimaszewska, Peter Stacey, Glenn A. Burley, John D. Harling, David J. Battersby, and Afjal H. Miah, RSC Med. Chem., 2025, 16, 1141-1150. 

173. . Georgina B. Armstrong, Glenn A. Burley, William Lewis, and Zahra Rattray, Mol. Pharmaceutics, 2024, 21, 6423-6432. 

172. . Francesco Rianjongdee, David Palmer, Stephen D. Pickett, Peter Pogany, Nicholas C. O. Tomkinson, and Darren V. S. Green, Chem. Inf. Model., 2024, 64, 4687-4699.

171. . Luke Chen, James D. F. Thompson, and Craig Jamieson, Chem. Eur. J., 2024, e202403128. 

170. . Laura C. Paterson, Philip G. Humphreys, Henry A. Kelly, and William J. Kerr, Drug Disc. Today, 2024, 29, 104162. 

169. . Georgina B. Armstrong, Alan Lewis, Vidhi Shah, Paul Taylor, Craig Jamieson, Glenn A. Burley, William Lewis, ad Zahra Rattray, ACS Pharmacol. Transl. Sci., 2024, 7, 2439-2451. 

168. . Georgina B. Armstrong, Vidhi Shah, Paula Sanches, Mitul Patel, Ricky Casey, Craig Jamieson, William J. Lewis, and Zahra Rattray, Comput. Struct. Biotechnol. J., 2024, 23, 2345-2357.

167. . Nathan M. L. Knight, James D. J. Thompson, John A. Parkinson, David M. Lindsay, Tell Tuttle, and William J. Kerr, Adv. Synth. Catal., 2024, 366, 2577-2586.

166. . Rebecca Stevens, James D. F. Thompson, Julie C. L. Fournier, Glenn A. Burley, David J. Battersby, and Afjal H. Miah, Chem. Soc. Rev., 2024, 53, 4838-4861.

165. . Cassie Pratley, Sabine Fenner, and John A. Murphy, Org. Lett., 2024, 26, 1287-1292.

164. . Thomas Grunshaw, Susanna H. Wood, Stephen Sproules, Andrew Parrott, Alison Nordon, Peter D. P. Shapland, Katherine M. P. Wheelhouse, and Nicholas C. O. Tomkinson, J. Org. Chem., 2024, 89, 7933-7945.

163. . Roderick P. Bunschoten, Frederik Peschke, Andrea Taladriz-Sender, Emma Alexander, Matthew J. Andrews, Alan R. Kennedy, Neal J. Fazakerley, Guy C. Lloyd Jones, Allan J. B. Watson, and Glenn A. Burley, J. Am. Chem. Soc., 2024, 146, 13558-13570.

162. . Chelsea D. Grace, Simon Nicolle, and John A. Murphy, Arkivoc, 2024, 202312115.

161. . Holly E. Bonfield, Colin M. Edge, Marc Reid, Alan R. Kennedy, David D. Pascoe, David M. Lindsay, and Damien Valette, Org. Lett., 2024, 26, 2857-2861.

160. . Seb Tyerman, Craig M. Robertson, and John A. Murphy, Org. Biomol. Chem., 2024, 22, 1023-1026.

159. . Kenneth F. Clark, Seb Tyerman, Laura Evans, Craig M. Roberson, and John A. Murphy, Org. Biomol. Chem., 2024, 22, 1018-1022.

158. . Thomas D. Fleetwood, William J. Kerr, and Joseph Mason, Chem. Eur. J., 2024, 30, e202303314.

157. . Joseph M. Anderson, Darren L. Poole, Gemma C. Cook, John A. Murphy, and Nicholas D. Measom, Chem. Eur. J., 2023, 30, e202304070.

156. . Aristea Anna Leventi, Henry J. Braddick, Kharmen Billimoria, Gregory Q. Wallace, Heidi Goenaga-Infante, Nicholas C. O. Tomkinson, Karen Faultds, and Duncan Graham, Chem. Commun., 2023, 29, 6395-6398.

155. . Sergej Maciuk, Susanna H. Wood, Vipulkumr K. Patel, Peter D. P. Shapland, and Nicholas C. O. Tomkinson, Chem. Eur. J., 2023, 29, e202204007.

154. . David J. Fallon, Alex Phillipou, Christopher J. Schofield, David House, Nicholas C. O. Tomkinson, and Jacob T. Bush, Biochem. J., 2023, 480, 1183-1197.

153. . Joseph Mason, Harry Wilders, David J. Fallon, Ross P. Thomas, Jacob T. Bush, Nicholas C. O. Tomkinson, and F. Rianjongdee, Digital Discovery, 2023, 2, 1894-1899.

152.  Brett Cosgrove, Emma K. Grant, Sophie Bertrand, Kenneth D. Down, Don O. Somers, John P. Evans, Nicholas C. O. Tomkinson, and Michael D. Barker, RSC Chem. Biol., 2023, 4, 1111-1122.

151. . Neville Murphy, William J. Tipping, Henry J. Braddick, Liam T. Wilson, Nicholas C. O. Tomkinson, Karen Faulds, Duncan Graham, and Pau Farras, Angew. Chem. Int. Ed., 2023, 62, e202311530.

150. . Kenneth F. Clark, Seb Tyerman, Laura Evans, Craig M. Robertson, David J. Nelson, Alan R. Kennedy, and John A. Murphy, J. Am. Chem. Soc., 2023, 145, 20849-20858.

149.   Erin Bradley, Lucia Fusani, Chun-wa Chung, Peter D. Craggs, Emmanuel H. Demont, Philip G. Humphreys, Darren J. Mitchell, Alex Phillipou, Inmaculada Rioja, Rishi R. Shah, Christopher R. Wellaway, Rab K. Prinjha, David S. Palmer, William J. Kerr, Marc Reid, Ian D. Wall, and Rosa Cookson, J. Med. Chem., 2023, 66, 15728-15749.

148. .  Karina Chan, Preethi Soundarya Sathyamurthi, Markus A. Queisser, Michael Mullin, Harry Shrives, Diane M. Coe, and Glenn A. Burley, Bioconjugate Chem., 2023, 34, 2049-2054.

147. . Rebecca Stevens, Enrique Bendito-Moll, David J. Battersby, Afjal H. Miah, Justyna M. Macina, Glenn A. Burley, and John D. Harling, J. Med. Chem., 2023, 66, 15437-15452.

146. . Marina Economidou, Nisha Mistry, Katherine M. P. Wheelhouse, and David M. Lindsay, Org. Process Res. Dev., 2023, 27, 1585-1615.

145. .  Elliot Davenport, Daniela E. Negru, Geoff Badman, David M. Lindsay, and William J. Kerr, ACS Catal., 2023, 13, 11541-11547.

144. .  Callum G. J. Hall, Helen F. Sneddon, Peter Pogany, David M. Lindsay, and William J. Kerr, Chem. Sci., 2023, 24, 6738-6755. 

143. . Claudine S. Greenwood, Meghan A. Wynosky-Dolfi, Allison M. Beal, and Lee M. Booty, Frontiers in Immunology, 2023, 14, 1173519.  DOI: 10.3389/fimmu.2023.1173519.

142. . Daniel J. Fowles, Rose G. McHardy, Abdullah Ahmad, and David S. Palmer, Digital Discovery, 2023, 2, 177-188.

141. . Daniel J. Fowles and David S. Palmer, Phys. Chem. Chem. Phys., 2023, 25, 6944-6954.

140. . Arron Aatkar, Aini Vuorinen, Oliver E. Longfield, Katharine E. Gilbert, Rachel Peltier-Heap, Craig D. Wagner, Francesca Zappacosta, Katrin Rittinger, Chun-wa Chung, David House, Nicholas C. O. Tomkinson, and Jacob T. Bush, ACS Chem. Biol., 2023, 18, 1926-1937.

139. . Henry J. Braddick, William J. Tipping, Liam T. Wilson, Harry S. Jaconelli, Emma K. Grant, Karen Faulds, Duncan Graham, and Nicholas C. O. Tomkinson, Anal. Chem., 2023, 95, 5369-5376.

138. . Sergej Macuik, Susanna H. Wood, Vipulkumar K. Patel, Peter D. P. Shapland, and Nicholas C. O. Tomkinson, Chem. Eur. J., 2023, 29, e202204007.

137. . Ross P. Thomas, Emma K. Grant, Eleanor R. Dickinson, Francesca Zappacosta, Lee J. Edwards, Michael M. Hann, David House, Nicholas C. O. Tomkinson, and Jacob T. Bush, RSC Med. Chem., 2023, 14, 671-679. 

136. .  Christopher M. Riley, Jessica M. L. Elwood, Martyn C. Henry, Irene Hunter, J. Daniel Lopez-Fernandez, Iain J. McEwan, and Craig Jamieson, Med. Res. Rev., 2023, 43, 1701-1747.

135. . Jason D. Williams, Stuart G. Leach, and William J. Kerr, Chem. Eur. J., 2023, 29, e202300403.  

134. . Joseph M. Anderson, Nicholas D. Measom, John A. Murphy, and Darren L. Poole, Org. Lett., 2023, 25, 2053-2057.

133.  Katharine E. Gilbert, Aini Vuorinen, Arron Aatkar, Peter Pogány, Jonathan Pettinger, Emma K. Grant, Joanna M. Kirkpatrick, Katrin Rittinger, David House, Glenn A. Burley, and Jacob T. Bush, ACS Chem. Biol., 2023, 18, 285-295.

132. . William J. Tipping, Liam T. Wilson, Connie An, Aristea A. Leventi, Alastair W. Wark, Corrina Wetherill, Nicholas C. O. Tomkinson, Karen Faults, and Duncan Graham, Chem. Sci., 2022, 13, 3468-3476.

131. .  Daniela Dimitrova, Connor McMahon, Alan R. Kennedy, John A. Parkinson, Stuart G. Leach, Lee T. Boulton, David D. Pascoe, and John A. Murphy, Tetrahedron, 2022, 128, 1331120.

130. . Philip G. Humphreys, Niall A. Anderson, Paul Bamborough, Andrew Baxter, Chun-wa Chung, Rosa Cookson, Peter D. Craggs, Toryn Dalton, Julie C. L. Fournier, Laurie J. Gordon, Heather F. Gray, Matthew W. Gray, Richard Gregory, David J. Hirst, Craig Jamieson, Katherine L. Jones, Hripsimee Kessedjian, David Lugo, Grant McGonagle, Vipulkumar K. Patel, Christopher Patten, Darren L. Poole, Rab K. Prinjha, Cesar Ramirez-Molina, Inmaculada Rioja, Gail Seal, Kayleigh A. J. Stafford, Rishi R. Shah, Daniel Tape, Natalie H. Theodoulou, Laura Tomlinson, Sabri Ukuser, Ian D. Wall, Natalie Wellaway, and Gemma White, J. Med. Chem., 2022, 65, 15174-15207.

129. .  Gaochao Tian, Steven R. Katchur, Yong Jiang, Jacques Briand, Michael Schaber , Constantine Kreatsoulas, Benjamin Schwartz, SaraThrall, Alicia M. Davis, Sam Duvall, Brett A. Kaufman, and William L. Rumsey, Sci. Rep., 2022, 12, 14685.

128.  Paul Shaw, Storm J. Hassell-Hart, Gayle E. Douglas, Andrew G. Malcolm, Alan R. Kennedy, Gemma V. White, Laura C. Paterson, and William J. Kerr, Org. Lett., 2022 24, 2750-2755. 

127. .  Andrew Jordan, Callum G. J. Hall, Lee R. Thorp, and Helen F. Sneddon, Chem. Rev., 2022, 122, 6749–6794.

126. .  Jonathan D. Bell, Iain Robb, and John A. Murphy, Chem. Sci., 2022, 13, 12921-12926.

125.   Emma Campbell, Andrea Taladriz-Sender, Olivia l. Paisley, Alan R. Kennedy, Jacob T. Bush, and Glenn A. Burley, J. Org. Chem., 2022 87, 4603-4616. 

124.  Cassie Pratley, Sabine Fenner, and John A. Murphy, Chem. Rev., 2022, 122, 8181–8260.

123.  Andrew Jordan, Callum G. J. Hall, Lee R. Thorp, and Helen F. Sneddon, Chem. Rev., 2022, 122, 6749-6794.

122.  Samuel D. L. Holman, Alfie G. Wills, Neal. J. Fazakerley, Darren L. Poole, Diane M. Coe, Leonard Berlouis, and Marc Reid, Chem. Eur. J., 2022, 28, e20210372.

121. Philip G. Humphreys, Stephen J. Atkinson, Paul Bamborough, Rino A. Bit, Chun-wa Chung, Peter D. Craggs, Leanne Cutler, Rob Davis, Alan Ferrie, GangLi Gong, Laurie J. Gordon, Matthew Gray, Lee A. Harrison, Thomas G. Hayhow, Andrea Haynes, Nick Henley, David J. Hirst, Ian D. Holyer, Matthew J. Lindon, Cerys Lovatt, David Lugo, Scott McCleary, Judit Molnar, Qendresa Osmani, Chris Patten, Alex Preston, Inmaculada Rioja, Jonathan T. Seal, Nicholas Smithers, Fenglai Sun, Dalin Tang, Simon Taylor, Natalie H. Theodoulou, Clare Thomas, Robert J. Watson, Christopher R. Wellaway, Linrong Zhu, Nicholas C. O. Tomkinson, and Rab K. Prinjha. J. Med. Chem., 2022,  2262–2287.

120.  Jonathan D. Bell and John A. Murphy, Chem. Soc. Rev., 2021, 50, 9540-9685.

119.  Jack Robertson, Marzuq A. Ungogo, Mustafa M. Aldfer, Leandro Lemgruber, Fergus S. McWhinnie, Bela E. Bode, Katherine L. Jones, Allan J. B. Watson, Harry P. de Koning, and Glenn A. Burley, ChemMedChem, 2021, 16, 3396-3401.

118.  Joseph M. Anderson, Nicholas D. Measom, John A. Murphy and Darren L. Poole. Angew. Chem. Int. Ed., 2021, 60, 24754-24769.

117.  Michael A. Clegg, Natalie H. Theodoulou, Paul Bamborough, Chun-wa Chung, Peter D. Craggs, Emmanuel H. Demont, Laurie J. Gordon, Gemma M. Liwicki, Alex Phillipou, Nicholas C. O. Tomkinson, Rab K. Prinjha, and Philip G. Humphreys. ACS Med. Chem. Lett., 2021, 12, 1308-1317.

116. . Peter Stacey, Hannah Lithgow, Xiao Lewell, Agnieszka Konopacka, Stephen Besley, Georgina Green, Ryan Whatling, Robert Law, Sascha R枚th, Gopal P. Sapkota, Ian E. D. Smith, Glenn A. Burley, John Harling, Andrew B. Benowitz, Markus A. Queisser, and Marcel Muelbaier. SLAS DISCOVERY: Advancing the Science of Drug Discovery, 2021, 6, 885-895.

115. , Daniel J. Fowles, David S. Palmer, Rui Guo, Sarah L. Price, John B. O. Mitchell, J. Chem. Theory Comput. 2021, 17, 3700-3709.

114. . Jack B. Washington, Michele Assante, Chunhui Yan, David R McKinney, Vanessa Juba, Andrew Leach, Sharon E Baillie, and Marc Reid. Chem. Sci., 2021, 12, 6949-6963.

113.   Rhys A. Lippa, David J. Battersby, John A. Murphy, and Tim N. Barrett.  J. Org. Chem., 2021, 86, 3583-3604.

112.   Blake J. Baker, William J. Kerr, David M. Lindsay, Vipulkumar K. Patel, and Darren L. Poole.  Green Chem., 2021, 23, 280-287.

111.   Brett Cosgrove, Kenneth Down, Sophie Bertrand, Nicholas C. O. Tomkinson, and Michael D. Barker.  Bioorg. Med. Chem. Lett., 2021, 33, Article No. 127752. 

110.   Youssef Shaalan, Lee Boulton, and Craig Jamieson.  Org. Process Res. Dev., 2020, 24, 2745-2751.

109. .  Simon C. C. Lucas, Stephen J. Atkinson, Paul Bamborough, Heather Barnett, Chun-wa Chung, Laurie Gordon, Darren J. Mitchell, Alexander Phillipou, Rab K. Prinjha, Robert J. Sheppard, Nicholas C. O. Tomkinson, Robert J. Watson, and Emmanuel H. Demont.  J. Med. Chem., 2020, 63, 5212-5241.

108. . .  Jonathan M. Curle, Marina C. Perieteanu, Phillip G. Humprhreys, Alan R. Kennedy, Nicholas C. O. Tomkinson.  Org. Lett., 2020, 22, 1659-1664.

107.   Andrew J. Smith, Daniela Dimitrova, Jude N. Arokianathar, Kenneth F. Clark, Darren L. Poole, Stuart G. Leach, and John A. Murphy.  Chem. Sci., 2020, 11, 12364-12370..

106. .  Connor A. Lawson, Andrew P. Dominey, Glynn D. Williams, and John A. Murphy, Chem. Commun., 2020, 56, 11445-11448.

105. . Simon Rohrbach, John A. Murphy, and Tell Tuttle.  J. Am. Chem. Soc., 2020, 142, 14871-14876.

104. . Luke Green, Keith Livingstone, Sophie Bertrand, Simon Peace, and Craig Jamieson.  Chem. Eur. J., 2020, 26, 14866-14870.

103. . Keith Livingstone, Sophie Bertrand, Alan R. Kennedy, and Craig Jamieson. Chem. Eur. J., 2020, 26, 10591-10597.

102. . Keith Livingstone, Sophie Bertrand, and Craig Jamieson. J. Org. Chem., 2020, 85, 7413-7423.

101. .  Sarah J. M. Patterson, Peter R. Clark, Glynn D. Williams, and Nicholas C. O. Tomkinson.  Tet. Lett., 2020, 61, article number 152483.

100.  Rhys Lippa, John Barrett, Sandeep Pal, James E. Rowedder, John A. Murphy, and Tim N. Barrett. Eur. J. Med. Chem., 2020, 208, article number 112719.

99.  Holly Bonfield, Damien Valette, David M. Lindsay, and Marc Reid, Chem. Eur. J., 2020, 27, 158-174.

98.   Emma. K. Grant, David J. Fallon, Michael M. Hann, Ken G. M. Fantom, Chad Quinn, Francesca Zappacosta, Roland S. Annan, Chun-wa Chung, Paul Bamborough, David P. Dixon, Peter Stacey, David House, Vipulkumar K. Patel, Nicholas C. O. Tomkinson, and Jacob Bush, Angew. Chem. Int. Ed., 2020, 59, 21096-21105.

97.  Christopher R. Wellaway, Paul Bamborough, Sharon G. Bernard, Chun-wa Chung, Peter D. Craggs, Leanne Cutler, Emmanuel H. Demont, John P. Evans, Laurie Gordon, Bhumika Karamshi, Antonia J. Lewis, Matthew J. Lindon, Darren J. Mitchell, Inmaculada Rioja, Peter E. Soden, Simon Taylor, Robert J. Watson, Rob Willis, James M. Woolven, Beata S. Wyspia艅ska, William J. Kerr, and Rab K. Prinjha, J. Med. Chem., 2020, 63, 9020-9044.

96.  Rhys A. Lippa, John A. Murphy, and Tim N. Barrett, Belstein J. Org. Chem., 2020, 16, 1617-1626.

95. . Alfie Wills, Darren L. Poole, Catherine M. Alder, and Marc Reid, ChemElectroChem, 2020, 7, 2771-2776.

94.  Michael Clegg, Paul Bamborough, Chun-Wa Chung, Peter D Craggs, Laurie J. Gordon, Paola Grandi, Melanie Leveridge, Matthew Lindon, Gemma Michele Liwicki, Anne-Marie Michon, Judit Molnar, Inmaculada Rioja, Peter Soden, Natalie Theodoulou, Thilo Werner, Nicholas C. O. Tomkinson, Rab K. Prinjha, and Philip G Humphreys, J. Med. Chem., 2020, 63, 5816-5840.

93. .  Andrew J. Smith, Daniela Dimitrova, Jude N. Arokainathar, Krystian Kolodziejczak, Allan Young, Mark Allison, Darren L. Poole, Stuart G. Leach, John A. Parkinson, Tell Tuttle, and John A. Murphy, Chem. Sci., 2020, 11, 3719-3726.

92.   Rishi R. Shah, Joanna M. Redmond, Andrei Mihut, Malini Menon, John P. Evans, John A. Murphy, Michelle A. Bartholomew, and Diane M. Coe, Bioorg. Med. Chem., 2020, article number 115326.

91. .  Peter R. Clark, Glynn D. Williams, Jerome F. Hayes, and Nicholas C. O. Tomkinson, Angew. Chem. Int. Ed., 2020, 59, 6740-6744.

90. . Oliver J. Turner, David J. Hirst, and John A. Murphy, Chem. Eur. J., 2020, 26, 3026-3029.

89. . Lucia Fusani, David S. Palmer, Don O. Somers, and Ian D. Wall, J. Chem. Inf. Model., 2020, 60, 1528-1539.

88.   Holly E. Bonfield, Kayleigh Mercer, Alba Diaz-Rodriguez, Gemma C. Cook, Blandine S. J. McKay, Pawel Slade, George M. Taylor, Wei Xiang Ooi, Jason D. Williams, Jack P. M. Roberts, John A. Murphy, Luca Schmermund, Wolfgang Kroutil, Tamara Mielke, Jared Cartwright, Gideon Grogan, and Lee J. Edwards, ChemPhotoChem, 2020, 4, 45-51.

87. . Keith Livingstone, Sophie Bertrand, Jenna Mowat, and Craig Jamieson.  Chem. Sci., 2019, 10, 10412-10416. 

86. .  Iain J. W. McKean, Joanna C. Sadler, Anibal Cuetos, Amina Frese, Luke D. Humphreys, Gideon Grogan, Paul A. Hoskisson, and Glenn A. Burley. Angew. Chem. Int. Ed., 2019, 58, 17583-17588.

85.   Emma K. Grant, David J. Fallon, Christian Eberl, Ken G. M. Fantom, Francesca Zappacosta, Cassie Messenger, Nicholas C. O. Tomkinson, and Jacob Bush, Angew. Chem. Int. Ed., 2019, 58, 17322-17327.

84. . Peter R. Clark, Glynn D. Williams, and Nicholas C. O. Tomkinson. Org. Biomol. Chem., 2019, 17, 7943-7955.

83.   Tim N. Barrett, Jonathan A. Taylor, Daniel Barker, Panayiotis A. Procopiou, James D.F. Thompson, John Barrett, Joelle Le, Sean M. Lynn, Peter Pogany, Cassie Pratley, John M. Pritchard, James A. Roper, James E. Rowedder, Robert J. Slack, Giovanni Vitulli, Simon J. F. Macdonald, and William J. Kerr, J. Med. Chem., 2019, 62, 7543-7556. 

82. .  Simon Rohrbach, Andrew J. Smith, Jia H. Pang, Darren L. Poole, Tell Tuttle, Shunsuke Chiba, and John A. Murphy, Angew. Chem. Int. Ed., 2019, 48, 16368-16388.

81. .  Christopher P. Tinworth, Hannah Lithgow, Lars Dittus, Zuni I. Bassi, Sophie E. Hughes, Marcel Muelbaier, Han Dai, Ian E. D. Smith, William J. Kerr, Glenn A. Burley, Marcus Bantscheff, and John D. Harling, ACS Chem. Biol., 2019, 14, 342-347.

80. .  David L. Cain, Callum McLaughin, John J. Molloy, Cameron Carpenter-Warren, Niall A. Anderson, and Allan J. B. Watson, Synlett, 2019, 30, 787-791.

79. .  Susanna H. Wood, Stephen Etridge, Alan R. Kennedy, Jonathan M. Percy, and David J. Nelson, Chem. Eur. J., 2019, 25, 5574-5585.

78. .  Julia F. Hyslop, Sarah L. Lovelock, Allan J. B. Watson, Peter W. Sutton, and Gheorghe-Doru Roiban, Journal of Biotechnology, 2019, 293, 56-65.

77. . Michael A. Clegg, Nicholas C. O. Tomkinson, Rab K. Prinjha, and P. Humpreys, ChemMedChem, 2019, 14, 362-385.

76. , Julia F. Hyslop, Sarah L. Lovelock, Peter W. Sutton, Kristin K. Brown, Allan J. B. Watson, and Gheorghe-Doru Roiban, Angew. Chem. Int. Ed., 2018, 57, 13821鈥�13824.

75. . John A. Murphy, Oliver Turner, David Hirst, and Eric Talbot, Chem. Eur. J., 2018, 24, 28658-18662.

74.   Joshua P. Barham, Samuel E. Dalton, Mark Allison, Ciuseppe Nocera, Allan Young, Matthew P. John, Thomas McGuire, Sebastien Campos, Tell Tuttle, and John A. Murphy, J. Am. Chem. Soc., 2018, 140, 11510-11518.

73.   Julien C. Vantourout, Ling Li, Enrique Bendito-Moll, Sonia Chabbra, Kenneth Arrington, Bela E. Bode, Albert Isidro-Llobet, John A. Kowalski, Mark G. Nilson, Katherine M. P. Wheelhouse, John L. Woodward, Shiping Xie, David C. Leitch, and Allan J. B. Watson, ACS Catal., 2018, 8, 9560-9566. 

72.  John J. Molloy, Jan B. Metternich, Constantin G. Daniliuc, Allan J. B. Watson, and Ryan Gilmour, Angew. Chem. Int. Ed., 2018, 57, 3168-3172.

71.  . Jason D. Williams, William J. Kerr, Stuart G. Leach, and David M. Lindsay, Angew. Chem. Int. Ed., 2018, 57, 12126-12130.

70. . Carla Alamillo-Ferrer, Jonathan M. Curle, Stuart C. Davidson, Simon C. C. Lucas, Stephen J. Atkinson, Matthew Campbell, Alan R. Kennedy, and Nicholas C. O. Tomkinson, J. Org. Chem. 2018. 83, 6728鈥�6740.

69. . Holly E. Bonfield, Jason D. Williams, Wei Xiang Ooi, Stuart G. Leach, William J. Kerr, Lee J. Edwards, ChemPhotoChem, 2018, 2, 938-944.

68.   Robert P. Law, Stephen J. Atkinson, Paul Bamborough, Chun-wa Chung, Emmanuel H. Demont, Laurie J. Gordon, Matthew Lindon, Rab K. Prinjha, Allan J. B. Watson, and David J. Hirst, J. Med. Chem., 2018, 61, 4317-4334.

67.  Robert J. Griffiths, Wei C. Kong, Stephen A. Richards, Glenn A. Burley, Michael C. Willis, and Eric P. Talbot, Chem. Sci., 2018, 9, 2295-2300.

66. . Lucia Fusani, Ian Wall, David Palmer, and Alvaro Cortes, Bioinformatics, 2018, 34, 1947鈥�1948.

65.   Samuel E. Dalton, Lars Dittus, Daniel A. Thomas, M谩ire A. Convery, Joao Nunes, Jacob T. Bush, John P. Evans, Thilo Werner, Marcus Bantscheff, John A. Murphy, and Sebastien Campos, J. Am. Chem. Soc., 2018, 140, 932-939. 

64. . Andrew J. Smith, Allan Young, Simon Rohrback, Erin F. O'Connor, Mark Allison, HongShuang Want, Darren L. Poole, Tell Tuttle, and John A. Murphy, Angew. Chem. Int. Ed., 2017, 56, 12747-13751.

63. . Florimond Cumine, Allan Young, Hans-Ulrich Reissig, Tell Tuttle, and John A. Murphy,  Eur. J. Org. Chem., 2017, 6867鈥�6871.

62. . Marie-Pierre Dreanic, Colin M. Edge, and Tell Tuttle, ACS Omega, 2017, 2, 5737-5747.

61. . Thomas A. Clohessy, Alastair Roberts, Eric S. Manas, Vipulkumar K. Patel, Niall A. Anderson, and Allan J. B. Watson, Org. Lett., 2017, 19, 6368-6371. 

60.   William J. Kerr, David M. Lindsay, Philippa K. Owens, Marc Reid, Tell Tuttle, and Sebastien Campos, ACS Catal., 2017, 7, 7182-7186. 

59. .  Helena S. Buchanan, Steven M. Pauff, Tilemachos D. Kosmidis, Andrea Taladriz-Sender, Olivia I. Rutherford, Marine Z. C. Hatit, Sabine Fenner, Allan J. B. Watson, and Glenn A. Burley, Org. Lett., 2017, 19, 3759-3762. 

58.   Afjal H. Miah, Aurelie C. Champigny, Rebecca H. Graves, Simon T. Hodgson, Jonathan M. Percy, and Panayiotis A. Procopiou, Bioorg. Med. Chem., 2017, 25, 5327-5340.

57. . Jonathan A. Spencer, Craig Jamieson, and Eric P. A. Talbot, Org. Lett., 2017, 19, 3891-3894.

56. . Michael Clegg, Nicholas C. O. Tomkinson, Rab K. Prinjah, and Philip G. Humphreys, Future Med. Chem., 2017, 9, 1579-1582.

55. . Lygia S. de Moraes, Darren Edwards, Alastair J. Florence, Andrea Johnston, Blair F. Johnston, Catriona A. Morrison, and Alan R. Kennedy, Cryst. Growth Des., 2017, 17 (6), pp 3277鈥�3286.

54. . Florimond Cumine, Shengze Zhou, Tell Tuttle, and John A. Murphy, Org. Biomol. Chem., 2017, 15, 3324-3336.

53. . Joanna C. Sadler, Luke D. Humpreys, Radka Snajdrova, and Glenn A. Burley, ChemBioChem, 2017, 18, 992-995.

52. . Julien C. Vantourout, Haralampos N. Miras, Albert Isidro-Llobet, Stephen Sproules, and Allan J. B. Watson, J. Am. Chem. Soc., 2017,  139,  4769鈥�4779.

51. . James N. Sanderson, Andrew P. Dominey and Jonathan M. Percy, Adv. Synth. Catal. 2017, 359, 1007-1017.

50. . C. P. Seath, J. W. B. Fyfe, J. J. Molloy and A. J. B. Watson, Synthesis, 2017, 49, 891-898.

49. . John J. Molloy, Thomas A. Clohessy, Craig Irving, Niall A. Anderson, Guy C. Lloyd-Jones and Allan J. B. Watson, Chem. Sci., 2017, 8, 1551-1559.

48. . James W. B. Fyfe, Neal J. Fazakerley and Allan J. B. Watson, Angew. Chem. Int. Ed., 2017, 56, 1249-1253.

47. . Robert J. Griffiths, Glenn A. Burley and Eric P. A. Talbot, Org. Lett., 2017, 19, 870-873.

46. . Simon A. Watson, Andrew J. Edwards and John A. Parkinson, Analytical Letters, 2017, 50, 161-172.

45. . Joanna C. Sadler, Chun-Wa Chung, Julie E. Mosley, Glenn A. Burley and Luke D. Humphreys, ACS Chem. Biol., 2017, 12, 374-379.

44. . Nicholas D. Measom, Kenneth D. Down, David J. Hirst, Craig Jamieson, Eric S. Manas, Vipulkumar K. Patel and Don O. Somers, ACS Med. Chem. Lett., 2017, 8, 43-48.

43. .  Philip G. Humphreys,  Paul Bamborough,  Chun-Wa Chung,  Peter D. Craggs,  Laurie J. Gordon,  Paola Grandi,  Thomas G. Hayhow,  Jameed Hussain,  Katherine L. Jones,  Matthew Lindon,  Anne-Marie Michon,  Jessica F. Renaux,  Colin J. Suckling,  David F. Tough and  Rab K. Prinjha, J. Med. Chem., 2017,&苍产蝉辫;60,&苍产蝉辫;695鈥�709.

42.  Groups. Joshua P. Barham, Matthew P. John, and John A. Murphy, J. Am. Chem. Soc., 2016, 138, 15482-15487.

41. . William J. Kerr, Richard J. Mudd, Philippa K. Owens, Marc Reid, Jack A. Brown and Sebastien Campos, J. Labelled Compd. Radiopharm., 2016, 59, 601-603.

40. . Augustin Amour, Nick Barton, Anthony W. J. Cooper, Graham Inglis, Craig Jamieson, Christopher N. Luscombe, David Perez, Simon Peace, Paul Rowland, Chris Tame, Sorif Uddin, Giovanni Vitulli, and Natalie Wellaway.  J. Med. Chem., 2016, 59. 7239-7251.

39. . Jonathan M. Percy, Helena Emerson, James W. B. Fyfe, Alan R. Kennedy, Sergej Maciuk, David Orr, Lucie Rathouska, Joanna M. Redmond and Peter G. Wilson, Chemistry 鈥� A European Journal , 2016, 22, 12166-12175.

38. . Carla Alamillo-Ferrer, Marianna Karabourniotis-Sotti, Alan R. Kennedy, Matthew Campbell and Nicholas C. O. Tomkinson, Org. Lett., 2016, 18, 3102鈥�3105.

37. . David Orr, Jonathan M. Percy and Zoe A. Harrison, Chem. Sci., 2016, 7, 6369-6380.

36. . Natalie H. Theodoulou, Nicholas C. O. Tomkinson, Rab K. Prinjha, and Philip G. Humphreys, Current Opinion in Chemical Biology, 2016, 33, 58-66.

35.  Joshua P. Barham, Graeme Coulthard, Katie J. Emery, Eswararao Doni, Florimond Cumine, Giuseppe Nocera, Matthew P John, Leonard E. A. Berlouis, Thomas M. McGuire, Tell Tuttle, and John A. Murphy, J. Am. Chem. Soc., 2016,  138 , 7402鈥�7410.

34. . Paul Bamborough, Heather A. Barnett, Isabelle Becher, Mark J. Bird, Chun-Wa Chung, Peter D. Craggs, Emmanuel H. Demont, Hawa Diallo, David J. Fallon, Laurie J. Gordon, Paola Grandi, Clare I. Hobbs, Edward Hooper-Greenhill, Emma J. Jones, Robert P. Law, Armelle Le Gall, David Lugo, Anne-Marie Michon, Darren J. Mitchell, Rab K. Prinjha, Robert J. Sheppard, Allan J. B. Watson, and Robert J. Watson, ACS Med. Chem. Lett., 2016,  7 , 552鈥�557.

33. . Aymeric  P. Colleville, Richard A. J. Horan, Sandrine Olazabal, and Nicholas C. O. Tomkinson, Org. Process Res. Dev., 2016, 20, 1283鈥�1296.

32. . Julien C Vantourout, Robert P. Law, Albert Isidro-Llobet, Stephen J. Atkinson, and Allan J. B. Watson, J. Org. Chem., 2016, 81, 3942-3950.

31. . Marine Z. C. Hatit, Joanna C. Sadler, Liam A. McLean, Benjamin C. Whitehurst, Ciaran P. Seath, Luke D. Humphreys, Robert J. Young, Allan J. B. Watson, and Glenn A. Burley, Org. Lett., 2016, 18, 1694-1697.

30. . J. A. Borthwick, N. Ancellin, S. M. Bertrand, R. P. Bingham, P. S. Carter, C.-W. Chung, I. Churcher, N. Dodic, C. N. Fournier, P. L. Francis, A. Hobbs, C. Jamieson, S. D. Pickett, S. E. Smith, D. O. Somers, C. Spitzfaden, C. J. Suckling, and R. J. Young, J. Med. Chem., 2016, 59, 2452-2467.

29. . Joshua P. Barham, Graeme Coulthard, Ryan G. Kane, Nathan Delgado, Matthew P. John, and John A. Murphy, Angew. Chem. Int. Ed., 2016, 55, 4492-4496.  

28. . L. Shukla, L. A. Ajram, M. Begg, B. Evans, R. H. Graves, S. T. Hodgson, S. M. Lynn, A. H. Miah, J. M. Percy, P. A. Procopiou, S. A. Richards, and R. J. Slack, Eur. J. Med. Chem., 2016, 115, 14-25.

27. . William J. Kerr, Richard J. Mudd, and Jack A. Brown, Chemistry 鈥� A European Journal, 2016, 22,&苍产蝉辫;4738鈥�4742.

26. . Greg M. Anderson, Iain Cameron, John A. Murphy and Tell Tuttle, RSC Adv., 2016, 6, 11335-11343.

25. . Natalie H. Theodoulou, Nicholas C. O. Tomkinson, Rab K. Prinjha and Philip G. Humphreys, ChemMedChem, 2016, 11, 477鈥�487.

24. . Robert J. Slack, Maryam Hafeji, Rebecca Rogers, Steve B. Ludbrook, John F. Marshall, David J. Flint, Susan Pyne, and Jane C. Denyer, Pharmacology, 2016, 97, 114鈥�125.

23.  Natalie H. Theodoulou, Paul Bamborough, Andrew J. Bannister, Isabelle Becher, Rino A. Bit, Ka H. Che, Chun-wa Chung, Antje Dittmann, Gerard Drewes, David H. Drewry, Laurie Gordon, Paola Grandi, Melanie Leveridge, Matthew Lindon, Anne-Marie. Michon, Judit Molnar, Samuel C. Robson, Nicholas C. O. Tomkinson, Tony Kouzarides, Rab K. Prinjha and Philip G. Humphreys, J. Med. Chem., 2015, 59, 1425-1439.

22. . Carla Alamillo-Ferrer, Stuart J. Davidson, Michael J. Rawling, Natalie H. Theodoulou, Matthew Campbell, Phillip G. Humphreys, Alan R. Kennedy, and Nicholas C. O. Tomkinson, Org. Lett., 2015, 17, 5132-5135.

21. . James W. B Fyfe and Allan J. B. Watson, Synlett, 2015, 26, 1139-1144.

20. . John J Molloy, Robert P. Law, James W. B. Fyfe, Ciaran P. Seath, David J. Hirst, and Allan J. B. Watson, Org. Biomol. Chem., 2015, 13, 3093-3102.

19. . James W. B. Fyfe, E. Valverde, Ciaran P. Seath, Alan R. Kennedy, Joanna M. Redmond, Niall A. Anderson, and Allan J. B. Watson,Chemistry 鈥� A European Journal, 2015, 21, 8951-8964.

18.  Calum W. Muir, Julien C. Vantourout, Albert Isidro-Llobet, Simon J. F. MacDonald, and Allan J. B. Watson, Org. Lett., 2015, 17, 6030-6033.

17.  Sophie M. Bertrand, Nicolas Ancellin, Benjamin Beaufils, Ryan P. Bingham, Jennifer A. Borthwick, Anne-Benedicte. Boullay, Eric Boursier, Paul S. Carter, Chun-wa. Chung, Ian Churcher, Nerina Dodic, Marie-Helene. Fouchet, Charlene Fournier, Peter L. Francis, Laura A. Gummer, Kenny Herry, Andrew Hobbs, Clare I. Hobbs, Paul Homes, Craig Jamieson, Edwige Nicodeme, Stephen D. Pickett, Iain H. Reid, Graham L. Simpson, Lisa A. Sloan, Sarah E. Smith, Donald O鈥橬. Somers, Claus Spitzfaden, Colin J. Suckling, Klara Valko, Yoshiaki Washio, and Robert J. Young, J. Med. Chem., 2015, 58, 7140-7163.

16.  John J. Molloy, Robert P. Law, James W. B. Fyfe, Ciaran P. Seath, David J. Hirst and Allan J. B. Watson, Org. Biomol. Chem., 2015, 13, 3093-3102.

15.  Joshua P. Barham, Matthew P. John, John A. Murphy, Beilstein J. Org. Chem., 2014, 10,&苍产蝉辫;2981鈥�2988.

14.  James W. B Fyfe, Ciaran P Seath, and Allan J. B Watson, Angew. Chem. Int. Ed., 2014, 53, 12077-12080.

13.  Shengze Zhou, Eswararao Doni, Greg M. Anderson, Ryan G. Kane, Scott W. MacDougall, Victoria M. Ironmonger, Tell Tuttle and John A. Murphy, J. Am. Chem. Soc., 2014, 136, 17818鈥�17826. 

12.  W. J. Kerr, R. J. Mudd, L. C. Paterson, and J. A. Brown, Chem. Eur. J., 2014, 20, 14604-14607.

11.  David Orr, Jonathan M. Percy, Tell Tuttle, Alan R. Kennedy and Zo毛 A. Harrison, Chem. Eur. J., 2014, 20, 14305鈥�14316.

10.  S. Stewart, R. Harris, and C. Jamieson, Synlett, 2014, 25, 2480-2484.

9.  A. P. Colleville, R. A. J. Horan, and N. C. O. Tomkinson, Org. Process Res. Dev., 2014, 18, 1128鈥�1136.

8.  A. H. Miah, H. Abas, M. Begg, B. J. Marsh, D. E. O鈥橣lynn, A. J. Ford, J. M. Percy, P. A. Procopiou, S. A. Richards, and S.-A. Rumley, Bioorg. Med. Chem., 2014, 22, 4298-4311.

7.  A. H. Miah, R. C. B. Copley, D. O'Flynn, J. M. Percy, and P. A. Procopiou, Org. Biomol. Chem., 2014, 12, 1779-1792.

6.  S. Zhou, G. M. Anderson, B. Mondal, E. Doni, V. Ironmonger, M. Kranz, T. Tuttle, and J. A. Murphy, Chem. Sci., 2014, 5 , 476-482.

5.  M. J. Rawling, J. H. Rowley, M. Campbell, A. R. Kennedy, J. A. Parkinson, and N. C. O. Tomkinson, Chem. Sci., 2014, 5, 1777-1785.

4. . J. D. Harling, A. M. Deakin, S. Campos, R. Grimley, L. Chaudry, C. Nye, O. Polyakova, C. M. Besant, N. Barton, D. Somers, J. Barrett, R. H. Graves, L. Hanns, W. J. Kerr, and R. Solari, J. Biol. Chem., 2013, 288, 28195-28206.

3.  D. Orr, A. Tolfrey, J. M. Percy, J. Frieman, Z. A. Harrison, M. Campbell-Crawford, and V. K. Patel, Chem. Eur. J., 2013, 19, 9655-9662.

2.  Sylvain Picon, Michael Rawling, Matthew Campbell and Nicholas C. O. Tomkinson, Org. Lett., 2012, 14, 6250-6253.

1.  N. A. Anderson, B. J. Fallon, E. Valverde, S. J. F. MacDonald, J. M. Pritchard, C. J. Suckling, and A. J. B. Watson, Synlett, 2012, 23, 2817-2821.

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